SCHEMBL1663077

SCHEMBL1663077

CN(C)c1ccc(NC(=O)CCCc2cc3cc(C(=O)O)ccc3[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
MAPT P10636 4/20 0.54
NPC1 O15118 2/20 0.54
MAPK1 P28482 2/20 0.54
RAB9A P51151 2/20 0.54
ALOX15 P16050 2/20 0.54
NFKB1 P19838 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54
MCL1 Q07820 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HDAC3 O15379 4/20 0.47
HDAC4 P56524 4/20 0.47
HDAC1 Q13547 4/20 0.47
HDAC7 Q8WUI4 4/20 0.47
HDAC2 Q92769 4/20 0.47
HDAC10 Q969S8 4/20 0.47
HDAC11 Q96DB2 4/20 0.47
HDAC8 Q9BY41 4/20 0.47
HDAC6 Q9UBN7 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663278 0.89 ALDH1A1 (0.53) ALDH1A1MAPTNPC1MAPK1RAB9A
SCHEMBL1663735 0.79 HRH3 (0.44) ALDH1A1CYP2C9HPGDHRH3POLB
SCHEMBL1663128 0.76 MTNR1A (0.56) ALDH1A1MAPTMAPK1ALOX15HRH3
SCHEMBL1663062 0.76 MTNR1A (0.44) ALDH1A1HPGDHRH3
SCHEMBL1663712 0.74 MTNR1A (0.48) ALDH1A1MAPTSMN1; SMN2HDAC3HDAC4
SCHEMBL6152137 0.74 HRH3 (0.53) ALDH1A1HPGDHRH3THRBGAA
SCHEMBL1663190 0.74 MTNR1A (0.40) SMN1; SMN2HDAC1HDAC2APPHRH3
SCHEMBL13369823 0.74 MTNR1A (0.51) ALDH1A1SMN1; SMN2HPGDHRH3THRB
SCHEMBL1663073 0.73 MAPT (0.48) ALDH1A1MAPTNPC1MAPK1RAB9A
SCHEMBL10985371 0.72 HRH3 (0.51) ALDH1A1MAPTMEN1KMT2AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2642994-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS Ligand Pharmaceuticals Incorporated (US) 2013-10-02 EP disclosed
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2012068406-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2012-05-24 WO disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed