SCHEMBL16633648

SCHEMBL16633648

Cc1ccc(S(=O)(=O)O)c(CCNCc2cccc(C#N)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 1/20 0.47
NOS1 P29475 3/20 0.43
HTR2A P28223 1/20 0.43
DPP7 Q9UHL4 1/20 0.41
IDH1 O75874 1/20 0.40
CNR1 P21554 1/20 0.38
MPO P05164 1/20 0.38
NR3C1 P04150 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA9 Q16790 1/20 0.37
ERCC1 P07992 1/20 0.37
ERCC4 Q92889 1/20 0.37
CYP19A1 P11511 1/20 0.37
NAMPT P43490 1/20 0.37
VNN1 O95497 1/20 0.36
TBXA2R P21731 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16634084 0.94 SCN8A (0.50) SCN8ANOS1HTR2ADPP7IDH1
SCHEMBL16633108 0.87 SCN8A (0.40) SCN8ANOS1IDH1CNR1NR3C1
SCHEMBL16633649 0.76 KCNN4 (0.37) IDH1TBXA2R
SCHEMBL16633107 0.75 TBXA2R (0.38) HTR2ACNR1NAMPTTBXA2R
SCHEMBL16634085 0.74 KCNN4 (0.35) IDH1TBXA2R
SCHEMBL16633106 0.72 GFER (0.45) TBXA2RKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL2964170 0.72 TBXA2R (0.40) NOS1IDH1TBXA2R
SCHEMBL18917603 0.71 TDP1 (0.40) CYP19A1
SCHEMBL1180196 0.71 GAA (0.41) KDM4EMAPTHPGDTSHRHSD17B10
SCHEMBL30823619 0.71 GAA (0.41) KDM4EMAPTHPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9238632-B2 3-cyanoanilinoalkylarylpiperazine derivative and use thereof in preparing drugs NHWA Pharma, Corporation (CN) 2016-01-19 US disclosed
US-20150105399-A1 3-CYANOANILINOALKYLARYLPIPERAZINE DERIVATIVE AND USE THEREOF IN PREPARING DRUGS SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2015-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105399-A1 3-CYANOANILINOALKYLARYLPIPERAZINE DERIVATIVE AND USE THEREOF IN PREPARING DRUGS HTR5A, HTR3C, HTR3A SCN8A 489/4885NOS1 1614/4885HTR2A 18/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.