SCHEMBL16634085

SCHEMBL16634085

Cc1ccc(S(=O)(=O)O)c(CCCN(C)c2cccc(C#N)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.35
KCNA5 P22460 1/20 0.35
NOS2 P35228 1/20 0.35
KCNJ6 P48051 1/20 0.35
KCNJ5 P48544 1/20 0.35
KCNJ3 P48549 1/20 0.35
PER2 O15055 1/20 0.35
CRY1 Q16526 1/20 0.35
CRY2 Q49AN0 1/20 0.35
TBXA2R P21731 3/20 0.35
SLC6A4 P31645 1/20 0.34
GFER P55789 1/20 0.34
IDH1 O75874 1/20 0.33
EPAS1 Q99814 2/20 0.33
NR1H3 Q13133 1/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
STAT3 P40763 1/20 0.33
PTPRS Q13332 1/20 0.33
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16633649 0.96 KCNN4 (0.37) KCNN4KCNA5NOS2KCNJ6KCNJ5
SCHEMBL16633106 0.87 GFER (0.45) KCNN4KCNA5PER2CRY1CRY2
SCHEMBL644417 0.77 CA12 (0.40) NOS2SLC6A4
SCHEMBL16633108 0.77 SCN8A (0.40) TBXA2RSLC6A4IDH1
SCHEMBL16634084 0.77 SCN8A (0.50) TBXA2RIDH1
SCHEMBL16633107 0.75 TBXA2R (0.38) TBXA2R
SCHEMBL16633648 0.74 SCN8A (0.47) TBXA2RIDH1
SCHEMBL816601 0.74 GAA (0.39)
SCHEMBL5718625 0.74 GAA (0.39)
SCHEMBL30723203 0.74 GAA (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9238632-B2 3-cyanoanilinoalkylarylpiperazine derivative and use thereof in preparing drugs NHWA Pharma, Corporation (CN) 2016-01-19 US disclosed
US-20150105399-A1 3-CYANOANILINOALKYLARYLPIPERAZINE DERIVATIVE AND USE THEREOF IN PREPARING DRUGS SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2015-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150105399-A1 3-CYANOANILINOALKYLARYLPIPERAZINE DERIVATIVE AND USE THEREOF IN PREPARING DRUGS HTR5A, HTR3C, HTR3A KCNN4 604/4885KCNA5 134/4885NOS2 1430/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.