SCHEMBL1663569

SCHEMBL1663569

O=C(O)CCc1nc2c[c]ccc2[nH]1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.64
KDM4E B2RXH2 3/20 0.55
APEX1 P27695 1/20 0.55
PRKAG1 P54619 3/20 0.54
PRKAA2 P54646 3/20 0.54
PRKAB1 Q9Y478 3/20 0.54
PRKAA1 Q13131 1/20 0.54
PARP1 P09874 2/20 0.50
PARP2 Q9UGN5 2/20 0.50
ALDH1A1 P00352 3/20 0.45
MAPT P10636 2/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
GAA P10253 1/20 0.40
S1PR1 P21453 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661454 0.88 CHRM1 (0.64) CHRM1KDM4EAPEX1PRKAG1PRKAA2
Procodazole SCHEMBL838841 0.78 CHRM1 (1.00) CHRM1KDM4EAPEX1PRKAG1PRKAA2
Procodazole SCHEMBL349966 0.78 CHRM1 (1.00) CHRM1KDM4EAPEX1PRKAG1PRKAA2
Procodazole SCHEMBL29404024 0.78 CHRM1 (1.00) CHRM1KDM4EAPEX1PRKAG1PRKAA2
SCHEMBL699318 0.78 RAB9A (0.67) CHRM1ALDH1A1MAPTGAAPOLB
SCHEMBL2565679 0.78 MAOB (0.43) CHRM1KDM4EALDH1A1MAPT
Procodazole SCHEMBL5413283 0.75 CHRM1 (0.91) CHRM1KDM4EAPEX1PRKAG1PRKAA2
SCHEMBL19330024 0.74 DDAH1 (0.58) GAAPOLBPKM
SCHEMBL1662293 0.74 CYP1A2 (0.41) CHRM1KDM4EAPEX1PRKAG1PRKAA2
SCHEMBL11217654 0.73 PRKAG1 (0.69) CHRM1KDM4EAPEX1PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2306994-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF Amgen, Inc (US) 2011-04-13 EP disclosed
WO-2009154775-A1 S1P1 RECEPTOR AGONISTS AND USE THEREOF AMGEN INC. (US) 2009-12-23 WO disclosed