SCHEMBL166364

SCHEMBL166364

O=C(O)COc1ccc(CO)cc1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.63
ALDH1A1 P00352 3/20 0.58
SMN1; SMN2 Q16637 1/20 0.56
FFAR1 O14842 1/20 0.56
NR4A1 P22736 1/20 0.56
APEX1 P27695 1/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
PTPN7 P35236 2/20 0.55
MAPT P10636 1/20 0.55
PTPN12 Q05209 1/20 0.55
TSHR P16473 2/20 0.51
PPARG P37231 2/20 0.51
PPARD Q03181 2/20 0.51
HSD17B10 Q99714 1/20 0.51
TBXAS1 P24557 2/20 0.51
PPARA Q07869 2/20 0.50
LTA4H P09960 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12646485 0.94 ALOX15 (0.57) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL1551092 0.91 FFAR1 (0.72) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL339492 0.87 ALOX15 (0.81) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL2439826 0.84 ALOX15 (0.59) ALOX15ALDH1A1SMN1; SMN2FFAR1MEN1
SCHEMBL4883406 0.83 PTPN7 (0.67) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL9832704 0.83 ALOX15 (0.63) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL2642068 0.83 ALOX15 (0.63) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
SCHEMBL15389920 0.83 NR4A1 (0.46) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1
Triclofenol SCHEMBL9654652 0.83 MCL1 (0.49) ALOX15ALDH1A1MAPTPPARD
SCHEMBL4781395 0.82 ALOX15 (0.61) ALOX15ALDH1A1SMN1; SMN2FFAR1NR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3447 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12577200-B2 High-throughput method to rapidly add chemical moieties to a small molecule library MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2026-03-17 US claimed
US-20250288651-A1 Therapeutic APAC Molecule Comprising Heparin Conjugated to a Plasma Protein APLAGON OY (FI) 2025-09-18 US claimed
EP-4247541-B1 METHODS OF MAKING AND USING PLATFORMS FOR PEPTIDE SYNTHESIS AND COMPOSITIONS THEREOF PEPTILOGICS INC (US) 2024-08-28 EP claimed
US-20240002431-A1 METHODS OF MAKING AND USING PLATFORMS FOR PEPTIDE SYNTHESIS AND COMPOSITIONS THEREOF PEPTILOGICS, INC. (US) 2024-01-04 US claimed
EP-4247541-A1 METHODS OF MAKING AND USING PLATFORMS FOR PEPTIDE SYNTHESIS AND COMPOSITIONS THEREOF Peptilogics, Inc. (US) 2023-09-27 EP claimed
CN-112759632-B Preparation method of Sylvestin 昆明龙津药业股份有限公司 2023-08-18 CN claimed
US-11446361-B2 Therapeutic APAC molecule comprising heparin conjugated to a plasma protein APLAGON OY (FI) 2022-09-20 US claimed
WO-2022109456-A1 METHODS OF MAKING AND USING PLATFORMS FOR PEPTIDE SYNTHESIS AND COMPOSITIONS THEREOF LEE FRANCIS (US) 2022-05-27 WO claimed
WO-2022060459-A1 HIGH-THROUGHPUT METHOD TO RAPIDLY ADD CHEMICAL MOIETIES TO A SMALL MOLECULE LIBRARY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2022-03-24 WO claimed
US-20220089537-A1 HIGH-THROUGHPUT METHOD TO RAPIDLY ADD CHEMICAL MOIETIES TO A SMALL MOLECULE LIBRARY MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2022-03-24 US claimed
EP-0305929-B1 Membranes with bound oligonucleotides and peptides MILLIPORE CORP (US) 1996-04-10 EP claimed
EP-0400920-B1 Solid phase multiple peptide synthesis APPLIED IMMUNESCIENCES (US) 1995-11-15 EP claimed
EP-0625996-A1 POLYETHYLENE OR POLYPROPYLENE GLYCOL CONTAINING POLYMER. CARLSBERG AS (DK) 1994-11-30 EP claimed
US-5352756-A Solid support for synthesis of peptides CARLSBERG A/S (DK) 1994-10-04 US claimed
EP-0608779-A1 Apparatus for peptide synthesis SHIMADZU CORPORATION (JP) 1994-08-03 EP claimed
WO-1993016118-A1 POLYETHYLENE OR POLYPROPYLENE GLYCOL CONTAINING POLYMER CARLSBERG A/S (DK) 1993-08-19 WO claimed
EP-0433345-A1 PEPTIDE SYNTHESIS METHOD AND SOLID SUPPORT FOR USE IN THE METHOD. RISOE FORSKNINGSCENTER (DK) 1991-06-26 EP claimed
US-4923901-A Membranes with bound oligonucleotides and peptides MILLIPORE CORPORATION (US) 1990-05-08 US claimed
WO-1990002749-A1 PEPTIDE SYNTHESIS METHOD AND SOLID SUPPORT FOR USE IN THE METHOD Forskningscenter Risø (DK) 1990-03-22 WO claimed
EP-0305929-A2 Membranes with bound oligonucleotides and peptides MILLIPORE CORPORATION (US) 1989-03-08 EP claimed