SCHEMBL1663701

SCHEMBL1663701

O=Cc1ccccc1N1CCC(CCO)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.45
MMP3 P08254 1/20 0.42
MMP8 P22894 1/20 0.42
PTPN1 P18031 1/20 0.41
AKR1C3 P42330 2/20 0.40
LTA4H P09960 1/20 0.40
ADRA1A P35348 4/20 0.39
ADRA1D P25100 3/20 0.39
ADRA1B P35368 3/20 0.39
TYMP P19971 2/20 0.38
CHRM2 P08172 5/20 0.38
CHRM1 P11229 5/20 0.38
CHRM3 P20309 5/20 0.38
CHRM4 P08173 5/20 0.38
DRD2 P14416 4/20 0.38
DRD3 P35462 4/20 0.38
CHRM5 P08912 4/20 0.38
DRD4 P21917 3/20 0.38
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663082 0.88 PTPN1 (0.51) CSF1RPTPN1LTA4HADRA1AADRA1D
SCHEMBL7484378 0.86 CHRM4 (0.37) PTPN1ADRA1AADRA1DADRA1BCHRM4
SCHEMBL29954495 0.81 MAPT (0.41) PTPN1LTA4HADRA1AADRA1DADRA1B
SCHEMBL2552593 0.81 MAPT (0.41) PTPN1LTA4HADRA1AADRA1DADRA1B
SCHEMBL6223691 0.79 KMT2A (0.41) CSF1RCHRM2CHRM1CHRM3CHRM4
SCHEMBL3084372 0.78 MEN1 (0.58) CSF1RMMP3MMP8PTPN1AKR1C3
SCHEMBL2481062 0.77 MAPT (0.55) ADRA1ACHRM2CHRM1DRD2DRD3
SCHEMBL3084371 0.77 NPC1 (0.59) CSF1RMMP3MMP8PTPN1AKR1C3
SCHEMBL7527672 0.76 CHRM4 (0.53) CSF1RCHRM4DRD2DRD3DRD4
SCHEMBL16814881 0.76 NCF1 (0.49) CSF1RMMP3MMP8PTPN1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9622991-B2 Hematopoietic growth factor mimetic small molecule compounds and their uses LIGAND PHARMACEUTICALS INC. (US) 2017-04-18 US disclosed
US-9144557-B2 Hematopoietic growth factor mimetic small molecule compounds and their uses LIGAND PHARMACEUTICALS INC. (US) 2015-09-29 US disclosed
US-20150252043-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES CITIBANK, N.A., AS ADMINISTRATIVE AGENT 2015-09-10 US disclosed
US-20140243324-A1 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2014-08-28 US disclosed
EP-2642994-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS Ligand Pharmaceuticals Incorporated (US) 2013-10-02 EP disclosed
US-20120295904-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2012-11-22 US disclosed
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2012068406-A2 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS LIGAND PHARMACEUTICALS INCORPORATED (US) 2012-05-24 WO disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140243324-A1 USE OF HEMATOPOIETIC GROWTH FACTOR MIMETICS HGF, EPOR, MPL CSF1R 8/4885MMP3 1980/4885MMP8 1058/4885
US-20150252043-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES MPL, CSF3R, HGF CSF1R 4/4885MMP3 2026/4885MMP8 412/4885
US-20120295904-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES MPL, CSF3R, HGF CSF1R 4/4885MMP3 2026/4885MMP8 412/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.