SCHEMBL16638946

SCHEMBL16638946

COCn1c(C)nc(C)c(OC)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
CYP1A2 P05177 5/20 0.35
CYP3A4 P08684 3/20 0.35
BRD4 O60885 1/20 0.33
HSD17B10 Q99714 4/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
USP2 O75604 1/20 0.33
MAPK1 P28482 1/20 0.33
ADORA2B P29275 1/20 0.33
CASP1 P29466 2/20 0.32
CASP7 P55210 2/20 0.32
TSHR P16473 2/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
KDM4E B2RXH2 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2610718 0.79 ADORA2B (0.33) ALDH1A1CYP1A2CYP3A4BRD4HSD17B10
SCHEMBL2116829 0.79 ADORA2B (0.33) ALDH1A1CYP1A2CYP3A4BRD4HSD17B10
SCHEMBL15177937 0.76 ADORA2B (0.31) ADORA2B
SCHEMBL9733254 0.63 ADORA2B (0.33) ALDH1A1CYP1A2CYP3A4HSD17B10CYP2C9
SCHEMBL13383886 0.61 ADORA2B (0.40) ALDH1A1CYP3A4HSD17B10ADORA2BKDM4E
SCHEMBL214654 0.59 ADORA2B (0.36) ALDH1A1ADORA2B
SCHEMBL12861937 0.58 KDM4E (0.32) BRD4HSD17B10KDM4EKMT2A
SCHEMBL3522549 0.57 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP3A4BRD4HSD17B10
SCHEMBL14112924 0.55 KDM4E (0.32) HSD17B10KDM4E
SCHEMBL19094969 0.55 ADORA2B (0.47) ALDH1A1CYP1A2CYP3A4CYP2C19ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2626350-B1 CYCLOPROPANE COMPOUND EISAI R&D MAN CO LTD (JP) 2015-04-15 EP disclosed