SCHEMBL9733254

SCHEMBL9733254

COCn1c(C)nc2nc(O)cnc2c1=O

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 1/20 0.33
LMNA P02545 1/20 0.32
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND2 P30279 1/20 0.30
CCND3 P30281 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
MAPK1 P28482 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2116829 0.69 ADORA2B (0.33) ADORA2BUSP2ALDH1A1CYP1A2CYP3A4
SCHEMBL16638946 0.63 ALDH1A1 (0.35) ADORA2BLMNAUSP2ALDH1A1CYP1A2
SCHEMBL2610718 0.63 ADORA2B (0.33) ADORA2BUSP2ALDH1A1CYP1A2CYP3A4
SCHEMBL9196786 0.61 HCAR2 (0.36) ALDH1A1
SCHEMBL12292807 0.60 KDM4E (0.31)
SCHEMBL9196781 0.59 KDM4E (0.37)
SCHEMBL9190063 0.59 PIK3CG (0.36) LMNAALDH1A1
SCHEMBL9190075 0.58 PIK3CG (0.36) LMNAALDH1A1
SCHEMBL9194837 0.57 CDC7 (0.38) ALDH1A1
SCHEMBL9196608 0.57 AKR1B1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5167949-A Antiallergic LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1992-12-01 US disclosed