SCHEMBL16639238

SCHEMBL16639238

CN1CCC(F)(F)/C(=C\C(=O)O)c2cc(F)ccc21

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.40
AVPR2 P30518 1/20 0.38
AVPR1A P37288 1/20 0.38
CDK9 P50750 11/20 0.36
NOTUM Q6P988 1/20 0.35
PER2 O15055 1/20 0.33
PARK7 Q99497 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16639237 0.85 TRPA1 (0.38) TRPA1AVPR2AVPR1ANOTUMPER2
SCHEMBL18926568 0.73 AVPR2 (0.38) TRPA1AVPR2AVPR1A
SCHEMBL16628454 0.72 ALK (0.34) TRPA1CDK9
SCHEMBL16628455 0.72 ALK (0.34) TRPA1CDK9
SCHEMBL16628531 0.71 LMNA (0.39)
SCHEMBL9028915 0.61 AVPR2 (0.51) AVPR2AVPR1A
SCHEMBL16723442 0.61 CCNT1 (0.36) CDK9
SCHEMBL23761222 0.61 ALDH1A1 (0.47) NOTUMPARK7
SCHEMBL14256267 0.61 ALDH1A1 (0.38) CDK9NOTUMPARK7
SCHEMBL16639240 0.61 CA1 (0.37) NOTUMPER2PARK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2860175-A1 METHOD FOR PRODUCING 4,4,7-TRIFLUORO-1,2,3,4-TETRAHYDRO-5H-1-BENZAZEPINE COMPOUND AND INTERMEDIATE FOR SYNTHESIS THEREOF Astellas Pharma Inc. (JP) 2015-04-15 EP disclosed