Adenosine

Adenosine

SCHEMBL1664893

Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O.OC[C@H]1O[C@@H](n2cnc3c(O)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 0.89

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3

The experimentally established mechanism targets of Adenosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 known ✓ P0DMS8 4/20 0.89
ADORA2A known ✓ P29274 1/20 0.89
ADORA2B known ✓ P29275 1/20 0.89
ADORA1 known ✓ P30542 1/20 0.89
DPP4 P27487 1/20 0.89
MEN1 O00255 1/20 0.89
SLC28A1 O00337 1/20 0.89
MAP3K7 O43318 1/20 0.89
SLC28A2 O43868 1/20 0.89
GAPDH P04406 1/20 0.89
MAPK1 P28482 1/20 0.89
STAT6 P42226 1/20 0.89
PI4KA P42356 1/20 0.89
KMT2A Q03164 1/20 0.89
SMN1; SMN2 Q16637 1/20 0.89
PI4K2B Q8TCG2 1/20 0.89
DOT1L Q8TEK3 1/20 0.89
SLC29A1 Q99808 1/20 0.89
PI4K2A Q9BTU6 1/20 0.89
SLC28A3 Q9HAS3 1/20 0.89

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Adenosine SCHEMBL13362239 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL4522263 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL19107495 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL23804425 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL1821276 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL23420216 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL406207 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL24538665 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL2228590 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7
Adenosine SCHEMBL2403819 0.94 ADORA3 (1.00) ADORA3DPP4MEN1SLC28A1MAP3K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117535350-A Gene therapy for age-related diseases and disorders 哈佛学院董事及会员团体 2024-02-09 CN disclosed
CN-109844124-B Gene therapy for age-related diseases and disorders 哈佛学院董事及会员团体 2023-10-03 CN disclosed
US-20230220443-A1 CHARACTERIZATION OF S-ADENOSYL-L-METHIONINE-CONSUMING ENZYMES WITH 1-STEP EZ-MTASE: A UNIVERSAL COUPLED-ASSAY NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-07-13 US disclosed
WO-2023111095-A2 ENGINEERED IMMUNE CELL KING'S COLLEGE LONDON (GB) 2023-06-22 WO disclosed
CN-116042482-A Lactobacillus avium and application thereof in preparation of products for treating or relieving hyperuricemia 中国农业大学 2023-05-02 CN disclosed
CN-110612353-A RNA targeting of mutations via inhibitory tRNAs and deaminases 加利福尼亚大学董事会 2019-12-24 CN disclosed
CN-109844124-A Methods of gene therapy for age-related diseases and disorders 哈佛学院董事及会员团体 2019-06-04 CN disclosed
WO-2018156464-A1 CHARACTERIZATION OF S-ADENOSYL-L-METHIONINE-CONSUMING ENZYMES WITH 1-STEP EZ-MTASE: A UNIVERSAL COUPLED-ASSAY ALBERT EINSTEIN COLLEGE OF MEDICINE, INC. (US) 2018-08-30 WO disclosed
EP-2306201-B1 Methods and compositions for assaying homocysteine GEN ATOMICS (US) 2014-10-08 EP disclosed
EP-1644741-B1 METHODS AND COMPOSITIONS FOR ASSAYING HOMOCYSTEINE GEN ATOMICS (US) 2011-08-31 EP disclosed
EP-2306201-A1 Methods and compositions for assaying homocysteine GENERAL ATOMICS (US) 2011-04-06 EP disclosed
EP-2235201-A1 METHODS AND COMPOSITIONS FOR ASSAYING HOMOCYSTEINE GENERAL ATOMICS (US) 2010-10-06 EP disclosed
WO-2009089106-A1 METHODS AND COMPOSITIONS FOR ASSAYING HOMOCYSTEINE GENERAL ATOMICS (US) 2009-07-16 WO disclosed
EP-1677665-A4 DETERMINATION OF IONS USING ION-SENSITIVE ENZYMES GEN ATOMICS (US) 2009-07-01 EP disclosed
EP-1677665-A2 DETERMINATION OF IONS USING ION-SENSITIVE ENZYMES GENERAL ATOMICS (US) 2006-07-12 EP disclosed
EP-1644741-A2 METHODS AND COMPOSITIONS FOR ASSAYING HOMOCYSTEINE GENERAL ATOMICS (US) 2006-04-12 EP disclosed
WO-2005027725-A2 DETERMINATION OF IONS USING ION-SENSITIVE ENZYMES GENERAL ATOMICS (US) 2005-03-31 WO disclosed
WO-2005008252-A2 METHODS AND COMPOSITIONS FOR ASSAYING HOMOCYSTEINE GENERAL ATOMICS (US) 2005-01-27 WO disclosed
WO-1999007877-A1 BIOSENSOR FOR DETECTING ADENOSINE THE UNIVERSITY COURT OF THE UNIVERSITY OF ST. ANDREWS (GB) 1999-02-18 WO disclosed
US-5583035-A FOR BLOCKING MESSENGER RNA AND SUPPRESSING VIRUS REPRODUCTION BAYER AKTIENGESELLSCHAFT (DE) 1996-12-10 US disclosed