SCHEMBL16655565

SCHEMBL16655565

O=c1cc(O)c2ccccc2n1Br

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.57
ALDH1A1 P00352 7/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
MAPT P10636 3/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
THRB P10828 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA9 Q16790 1/20 0.39
CYP2C19 P33261 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
NQO2 P16083 2/20 0.38
HTT P42858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1523070 0.77 KDM4E (0.57) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL835056 0.77 KDM4E (0.65) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL3582572 0.77 KDM4E (0.57) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL2266248 0.77 KDM4E (0.57) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL11828702 0.75 KDM4E (0.55) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL4190262 0.74 ALDH1A1 (0.55) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL11826562 0.74 KDM4E (0.50) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL11826850 0.74 KDM4E (0.54) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL8076374 0.73 KDM4E (0.57) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL9535544 0.73 KDM4E (1.00) KDM4EALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057422-A1 QUINOLINYL MODULATORS OF ROR(GAMMA)T Janssen Pharmaceutica NV (BE) 2016-08-24 EP disclosed
WO-2015057626-A1 QUINOLINYL MODULATORS OF RORyT JANSSEN PHARMACEUTICA NV (BE) 2015-04-23 WO disclosed