SCHEMBL16655883

SCHEMBL16655883

O=C(COc1ccc(Cl)cc1)Nc1ccccc1C(=O)OBr

nearest known ligand 0.74

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.74
RAB9A P51151 5/20 0.74
TSHR P16473 3/20 0.62
MAPK10 P53779 2/20 0.62
ALDH1A1 P00352 1/20 0.62
HSD17B10 Q99714 1/20 0.62
L3MBTL1 Q9Y468 2/20 0.62
LMNA P02545 1/20 0.62
MAPT P10636 1/20 0.62
HPGD P15428 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.61
TP53 P04637 1/20 0.61
HCAR2 Q8TDS4 1/20 0.56
KMT2A Q03164 1/20 0.56
POLB P06746 3/20 0.56
NPSR1 Q6W5P4 1/20 0.54
SENP2 Q9HC62 1/20 0.53
SENP1 Q9P0U3 1/20 0.53
TDP1 Q9NUW8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4293558 0.88 ALDH1A1 (0.80) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL4912964 0.85 NPC1 (0.80) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL6720448 0.81 NPC1 (0.73) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL14960451 0.79 MAPT (0.71) NPC1RAB9ATSHRALDH1A1L3MBTL1
SCHEMBL4908172 0.77 ALDH1A1 (0.84) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL5696432 0.75 ALDH1A1 (0.80) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL12555378 0.75 NPC1 (0.64) NPC1RAB9ATSHRALDH1A1L3MBTL1
SCHEMBL5696463 0.75 ALDH1A1 (0.85) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL6032429 0.75 HCAR2 (0.81) NPC1RAB9ATSHRMAPK10ALDH1A1
SCHEMBL4915695 0.75 HCAR2 (0.76) NPC1RAB9ATSHRMAPK10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3083561-A1 HETEROARYL LINKED QUINOLINYL MODULATORS OF RORYT Janssen Pharmaceutica N.V. (BE) 2016-10-26 EP disclosed
WO-2015057200-A1 HETEROARYL LINKED QUINOLINYL MODULATORS OF RORϒT JANSSEN PHARMACEUTICA NV (BE) 2015-04-23 WO disclosed