SCHEMBL6720448

SCHEMBL6720448

O=C(COc1ccc(Cl)cc1)Nc1ccccc1C(=O)C(F)(F)F

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.73
RAB9A P51151 5/20 0.73
L3MBTL1 Q9Y468 2/20 0.60
LMNA P02545 1/20 0.60
MAPT P10636 1/20 0.60
HPGD P15428 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.57
TP53 P04637 1/20 0.57
POLB P06746 2/20 0.55
HCAR2 Q8TDS4 2/20 0.55
KMT2A Q03164 2/20 0.55
TSHR P16473 2/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPK10 P53779 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NPSR1 Q6W5P4 1/20 0.53
KDM4E B2RXH2 1/20 0.53
MLYCD O95822 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8368918 0.84 NPC1 (0.53) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL4912964 0.84 NPC1 (0.80) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL4293558 0.82 ALDH1A1 (0.80) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL16655883 0.81 NPC1 (0.74) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL14960451 0.78 MAPT (0.71) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL28316072 0.77 ALDH1A1 (0.60) NPC1RAB9ALMNAMAPTHPGD
SCHEMBL6804609 0.76 CYP1A2 (0.57) NPC1RAB9AL3MBTL1SMN1; SMN2TSHR
SCHEMBL8590044 0.75 HDAC3 (0.47) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL12555378 0.74 NPC1 (0.64) NPC1RAB9AL3MBTL1LMNAMAPT
SCHEMBL6032429 0.74 HCAR2 (0.81) NPC1RAB9AL3MBTL1SMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040087491-A1 Electrophilic ketones for the treatment of herpesvirus infections FLYNN DANIEL L (US) 2004-05-06 US claimed
US-20030119721-A1 Electrophilic ketones for the treatment of herpesvirus infections G. D. SEARLE & CO., CORPORATE PATENT DEPARTMENT 2003-06-26 US claimed
EP-0888322-B1 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS SEARLE & CO (US) 2002-09-18 EP claimed
EP-0888322-A2 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS G.D. SEARLE & CO. (US) 1999-01-07 EP claimed
WO-1997034566-A2 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS G.D. SEARLE & CO. (US) 1997-09-25 WO claimed
US-20040087491-A1 Electrophilic ketones for the treatment of herpesvirus infections FLYNN DANIEL L (US) 2004-05-06 US disclosed
US-6673788-B2 CONTAINING 2,2,2-TRIFLUORO-1-OXOETHYL GROUPS G. D. SEARLE & CO. 2004-01-06 US disclosed
US-6673784-B1 HALOSUBSTITUTED ACETOPHENONES AS SELECTIVE HERPESVIRUS PROTEASE INHIBITORS G. D. SEARLE & CO. 2004-01-06 US disclosed
US-20030119721-A1 Electrophilic ketones for the treatment of herpesvirus infections G. D. SEARLE & CO., CORPORATE PATENT DEPARTMENT 2003-06-26 US disclosed
EP-0888322-B1 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS SEARLE & CO (US) 2002-09-18 EP disclosed
EP-0888322-A2 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS G.D. SEARLE & CO. (US) 1999-01-07 EP disclosed
WO-1997034566-A2 ELECTROPHILIC KETONES FOR THE TREATMENT OF HERPESVIRUS INFECTIONS G.D. SEARLE & CO. (US) 1997-09-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087491-A1 Electrophilic ketones for the treatment of herpesvirus infections KHK, HCK, PBK NPC1 1523/4885RAB9A 1684/4885L3MBTL1 2040/4885
US-20030119721-A1 Electrophilic ketones for the treatment of herpesvirus infections KHK, HCK, PBK NPC1 1523/4885RAB9A 1684/4885L3MBTL1 2040/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.