SCHEMBL16655976

SCHEMBL16655976

O=C1N=CC(O)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
IDO1 P14902 2/20 0.36
PARP3 Q9Y6F1 1/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
ALOX15 P16050 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP2D6 P10635 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PKM P14618 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18954022 0.76 ALDH1A1 (0.36) ALDH1A1MEN1POLBKMT2AALOX15
SCHEMBL10372679 0.74 POLB (0.40) ALDH1A1MEN1POLBKMT2AEDNRB
SCHEMBL4685836 0.73 ALDH1A1 (0.46) ALDH1A1PARP3MEN1POLBKMT2A
SCHEMBL6080166 0.71 EDNRB (0.41) ALDH1A1MEN1POLBKMT2AEDNRB
SCHEMBL3616941 0.70 MAOA (0.36) MEN1KMT2AMAOAMAOB
SCHEMBL5223009 0.69 HTR6 (0.42) ALDH1A1HDAC8MAOB
SCHEMBL6607488 0.68 ALDH1A1 (0.39) ALDH1A1IDO1PARP3MEN1POLB
SCHEMBL2933046 0.68 GABRP (0.37) ALDH1A1MEN1POLBKMT2AALOX15
SCHEMBL6314591 0.68 MEN1 (0.40) ALDH1A1IDO1PARP3MEN1POLB
SCHEMBL3421519 0.67 ALDH1A1 (0.36) ALDH1A1MEN1POLBKMT2AEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057586-A1 BROMODOMAIN INHIBITORS Celgene Quanticel Research, Inc. (US) 2016-08-24 EP disclosed
WO-2015058160-A1 BROMODOMAIN INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2015-04-23 WO disclosed