SCHEMBL16656773

SCHEMBL16656773

COc1ccc(C(C)N(CC(=O)O)CC(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.51
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
FFAR1 O14842 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
LDHA P00338 1/20 0.45
KMT2A Q03164 3/20 0.44
ATM Q13315 1/20 0.44
MEN1 O00255 2/20 0.44
PTGS2 P35354 3/20 0.44
PTGS1 P23219 2/20 0.44
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 2/20 0.44
CDC42 P60953 1/20 0.44
RAC1 P63000 1/20 0.44
CYP1A2 P05177 1/20 0.44
TSHR P16473 1/20 0.44
SLC22A6 Q4U2R8 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16656762 1.00 ALOX5 (0.51) ALOX5KEAP1NFE2L2FFAR1L3MBTL1
SCHEMBL16656812 1.00 ALOX5 (0.51) ALOX5KEAP1NFE2L2FFAR1L3MBTL1
SCHEMBL29330579 0.85 ALOX5 (0.50) ALOX5KEAP1NFE2L2FFAR1L3MBTL1
SCHEMBL24495053 0.82 L3MBTL1 (0.46) ALOX5L3MBTL1KMT2AMEN1TSHR
SCHEMBL16656809 0.80 ALOX5 (0.52) ALOX5
SCHEMBL21798487 0.76 ALOX5 (0.54) ALOX5KMT2AMEN1PTGS2PTGS1
SCHEMBL21798482 0.76 ALOX5 (0.54) ALOX5KMT2AMEN1PTGS2PTGS1
SCHEMBL18783512 0.75 TAS1R3 (0.40) ALOX5PTGS2TSHRRAB9AALDH1A1
SCHEMBL5317085 0.75 HTT (0.55) FFAR1L3MBTL1LDHAKMT2AATM
SCHEMBL27590253 0.75 PDE4B (0.50) ALOX5FFAR1L3MBTL1LDHAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210009508-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates NATIONAL SCIENCE FOUNDATION 2021-01-14 US disclosed
US-10752577-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2020-08-25 US disclosed
US-20190315676-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2019-10-17 US disclosed
US-10239824-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2019-03-26 US disclosed
US-20170158614-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES NATIONAL SCIENCE FOUNDATION 2017-06-08 US disclosed
US-9388131-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2016-07-12 US disclosed
US-20150329567-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2015-11-19 US disclosed
US-9012658-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2015-04-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150329567-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885
US-10752577-B2 Automated synthesis of small molecules using chiral, non-racemic boronates BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885
US-20170158614-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885
US-20190315676-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885
US-10239824-B2 Automated synthesis of small molecules using chiral, non-racemic boronates BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885
US-20210009508-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates BTD, POLL, POLR1A ALOX5 1847/4885KEAP1 3703/4885NFE2L2 4679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.