SCHEMBL1668495

SCHEMBL1668495

COc1ccc(CCOCCC(=O)O)cc1C1(c2ccccc2)CCN(C)CC1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 13/20 0.56
CHRM1 P11229 12/20 0.56
CHRM3 P20309 10/20 0.56
SIGMAR1 Q99720 2/20 0.41
EBPL Q9BY08 1/20 0.37
SLC22A1 O15245 1/20 0.37
SLC6A4 P31645 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670735 0.90 CHRM5 (0.46) CHRM5CHRM1CHRM3SIGMAR1
SCHEMBL12801191 0.89 CHRM5 (0.46) CHRM5CHRM1CHRM3SLC22A1SLC6A4
SCHEMBL1668671 0.84 FFAR4 (0.44) CHRM5CHRM1CHRM3
SCHEMBL1668720 0.83 CHRM5 (0.43) CHRM5CHRM1CHRM3SLC22A1SLC6A4
SCHEMBL12800795 0.83 CHRM5 (0.45) CHRM5CHRM1CHRM3SIGMAR1SLC22A1
SCHEMBL1668281 0.81 CHRM5 (0.39) CHRM5CHRM1CHRM3SIGMAR1ADRA1A
SCHEMBL12800404 0.80 CHRM5 (0.40) CHRM5CHRM1CHRM3OPRM1
SCHEMBL12801208 0.80 FFAR4 (0.47) CHRM5CHRM1CHRM3SIGMAR1
SCHEMBL1668325 0.79 OPRM1 (0.42) CHRM5CHRM1CHRM3OPRM1OPRD1
SCHEMBL1668476 0.78 CYP2D6 (0.46) CHRM5CHRM1CHRM3OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed