SCHEMBL1668720

SCHEMBL1668720

CN1CCC(c2ccccc2)(c2cc(CCCOCCC(=O)O)ccc2O)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 9/20 0.43
CHRM3 P20309 9/20 0.43
CHRM1 P11229 8/20 0.43
OPRM1 P35372 4/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC22A1 O15245 1/20 0.38
ADRA1A P35348 1/20 0.38
KCNH2 Q12809 1/20 0.38
S1PR5 Q9H228 3/20 0.38
S1PR1 P21453 3/20 0.37
S1PR3 Q99500 2/20 0.37
DRD4 P21917 1/20 0.37
RXRA P19793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801191 0.94 CHRM5 (0.46) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL1668599 0.91 RXRA (0.38) CHRM5CHRM3CHRM1OPRM1SLC6A4
SCHEMBL1668322 0.90 S1PR1 (0.40) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL1668671 0.87 FFAR4 (0.44) CHRM5CHRM3CHRM1S1PR5S1PR1
SCHEMBL12800404 0.85 CHRM5 (0.40) CHRM5CHRM3CHRM1OPRM1S1PR5
SCHEMBL1668325 0.84 OPRM1 (0.42) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL12800415 0.84 CHRM5 (0.38) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL1668281 0.83 CHRM5 (0.39) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL1668495 0.83 CHRM5 (0.56) CHRM5CHRM3CHRM1OPRM1OPRD1
SCHEMBL1668476 0.83 CYP2D6 (0.46) CHRM5CHRM3CHRM1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed