SCHEMBL1668671

SCHEMBL1668671

CN1CCC(c2ccccc2)(c2cc(CCCOCCC(=O)O)ccc2OCc2ccccc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 3/20 0.44
CHRM5 P08912 4/20 0.43
CHRM1 P11229 4/20 0.43
CHRM3 P20309 4/20 0.43
FFAR1 O14842 2/20 0.42
PTGER1 P34995 1/20 0.39
PTGER4 P35408 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGER2 P43116 1/20 0.39
S1PR5 Q9H228 4/20 0.38
S1PR1 P21453 3/20 0.38
S1PR3 Q99500 2/20 0.38
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
APP P05067 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670735 0.95 CHRM5 (0.46) FFAR4CHRM5CHRM1CHRM3FFAR1
SCHEMBL1668720 0.87 CHRM5 (0.43) CHRM5CHRM1CHRM3S1PR5S1PR1
Hydrochloric Acid SCHEMBL1668222 0.86 FFAR1 (0.43) FFAR4FFAR1PTGER1PTGER4PTGER3
SCHEMBL12801208 0.85 FFAR4 (0.47) FFAR4CHRM5CHRM1CHRM3FFAR1
SCHEMBL1668495 0.84 CHRM5 (0.56) CHRM5CHRM1CHRM3
SCHEMBL1669343 0.82 OPRD1 (0.40) FFAR4CHRM5CHRM1CHRM3FFAR1
SCHEMBL12800403 0.82 OPRD1 (0.46) FFAR4
SCHEMBL12801191 0.81 CHRM5 (0.46) CHRM5CHRM1CHRM3APP
SCHEMBL1668599 0.78 RXRA (0.38) FFAR4CHRM5CHRM1CHRM3FFAR1
SCHEMBL1668322 0.78 S1PR1 (0.40) CHRM5CHRM1CHRM3S1PR5S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed