SCHEMBL1669126

SCHEMBL1669126

CC(=O)/C=C(/CC(C)=O)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
TSHR P16473 1/20 0.46
KDM6B O15054 1/20 0.36
KDM5C P41229 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
PHF8 Q9UPP1 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
MGAM O43451 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
HTT P42858 1/20 0.32
GRIK1 P39086 1/20 0.31
GRIK2 Q13002 1/20 0.31
LMNA P02545 1/20 0.31
SLC15A2 Q16348 1/20 0.31
ALDH1A1 P00352 2/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14478054 0.85 KDM4E (0.65) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL10071805 0.85 KDM4E (0.65) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL819099 0.85 TSHR (0.65) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL2622343 0.85 TSHR (0.65) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL11949181 0.82 MGAM (0.36) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL24180793 0.81 KDM4E (0.43) KDM4ETSHRKDM6BKDM5CEGLN1
SCHEMBL12989964 0.81 KDM4E (0.43) KDM4ETSHRGRIK1GRIK2LMNA
SCHEMBL12576175 0.81 KDM4E (0.43) KDM4ETSHRALDH1A1
SCHEMBL23760642 0.79 KDM4E (0.41) KDM4ETSHRLMNA
SCHEMBL13712337 0.79 KDM4E (0.41) KDM4ETSHRKDM6BKDM5CEGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046062-A1 USE OF PRODRUGS TO AVOID GI MEDIATED ADVERSE EVENTS SHIRE, LLC (US) 2012-04-12 WO disclosed
WO-2010112942-A1 NOVEL DICARBOXYLIC ACID LINKED AMINO ACID AND PEPTIDE PRODRUGS OF OPIOIDS AND USES THEREOF SHIRE LLC (US) 2010-10-07 WO disclosed
EP-2230312-A1 Probe compound for detecting and isolating enzymes and means and methods using the same Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2010-09-22 EP disclosed