SCHEMBL16693236

SCHEMBL16693236

O=Cc1ccc2c(C(F)(F)F)csc2c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.41
CYP2A6 P11509 3/20 0.39
CYP17A1 P05093 1/20 0.36
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
PTGS2 P35354 1/20 0.32
RAB9A P51151 1/20 0.32
ERN1 O75460 1/20 0.32
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16693190 0.80 KDM4E (0.37) CYP17A1ALDH1A1KDM4E
SCHEMBL16693235 0.80 APP (0.33) CYP17A1
SCHEMBL16693150 0.77 CYP2A6 (0.42) KIF11CYP2A6ALDH1A1KDM4EPTGS2
SCHEMBL3046361 0.75 CYP2A6 (0.43) KIF11CYP2A6ALDH1A1KDM4EPTGS2
SCHEMBL17345173 0.74 KIF11 (0.53) KIF11CYP2A6AKR1C3AKR1C2ALDH1A1
SCHEMBL16693081 0.74 CYP2A6 (0.42) KIF11CYP2A6CYP17A1ALDH1A1KDM4E
SCHEMBL18791161 0.74 LMNA (0.38) KIF11CYP17A1KDM4E
SCHEMBL3407569 0.74 CYP2A6 (0.39) CYP2A6CYP17A1MAOB
SCHEMBL14093011 0.71 KIF11 (0.45) KIF11CYP17A1ALDH1A1KDM4E
SCHEMBL472408 0.70 KIF11 (0.56) KIF11CYP2A6AKR1C3AKR1C2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed