SCHEMBL16701948

SCHEMBL16701948

O=c1[nH]c2cccc(C3CCN(Cc4ccc(OC5CCN(C6CCC6)CC5)cc4)CC3)c2o1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 16/20 0.40
KCNH2 Q12809 4/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR1A P08908 1/20 0.39
DRD2 P14416 1/20 0.39
ADRB2 P07550 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16712648 0.87 HRH3 (0.43) HRH3KCNH2HTR1ADRD2
SCHEMBL16702159 0.87 MAOA (0.41) HRH3MAOAMAOBHTR1ADRD2
SCHEMBL16703990 0.86 MAOA (0.39) HRH3MAOAMAOBHTR1ADRD2
SCHEMBL16702411 0.86 KCNH2 (0.45) HRH3KCNH2MAOAMAOBADRB2
SCHEMBL16701857 0.86 DRD2 (0.55) HTR1ADRD2
SCHEMBL16702060 0.82 HRH3 (0.58) HRH3KMT2A
SCHEMBL16701815 0.81 GPR119 (0.43) KCNH2HTR1ADRD2ADRB2MEN1
SCHEMBL16712642 0.79 HRH3 (0.55) HRH3
SCHEMBL16701992 0.76 HRH3 (0.53) HRH3HTR1ADRD2
SCHEMBL16712645 0.75 DRD2 (0.63) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069110-A1 MULTIPLE D2 A(NTA)GONISTS/H3 ANTAGONISTS FOR TREATMENT OF CNS-RELATED DISORDERS AAPA B.V. (NL) 2015-05-14 WO disclosed