SCHEMBL16702159

SCHEMBL16702159

O=c1[nH]c2cccc(C3CCN(Cc4ccc(OC5CCNCC5)cc4)CC3)c2o1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.41
MAOB P27338 4/20 0.41
HRH1 P35367 1/20 0.41
HRH3 Q9Y5N1 5/20 0.41
HTR1A P08908 7/20 0.41
DRD2 P14416 7/20 0.41
OPRM1 P35372 1/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
UTS2R Q9UKP6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16703990 0.87 MAOA (0.39) MAOAMAOBHRH3HTR1ADRD2
SCHEMBL16702411 0.87 KCNH2 (0.45) MAOAMAOBHRH3GAA
SCHEMBL16701948 0.87 HRH3 (0.40) MAOAMAOBHRH3HTR1ADRD2
SCHEMBL16702375 0.86 HTR1A (0.39) HTR1ADRD2UTS2R
SCHEMBL16701987 0.85 DRD2 (0.59) HTR1ADRD2
SCHEMBL16701815 0.83 GPR119 (0.43) HTR1ADRD2
SCHEMBL16702746 0.81 MBTD1 (0.43) HRH3HTR1ADRD2GAA
SCHEMBL16701992 0.79 HRH3 (0.53) HRH3HTR1ADRD2
SCHEMBL2450534 0.77 HTR2C (0.47) HTR1A
SCHEMBL16704219 0.76 MAOB (0.43) MAOAMAOBHRH3HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069110-A1 MULTIPLE D2 A(NTA)GONISTS/H3 ANTAGONISTS FOR TREATMENT OF CNS-RELATED DISORDERS AAPA B.V. (NL) 2015-05-14 WO disclosed
WO-2015069110-A1 MULTIPLE D2 A(NTA)GONISTS/H3 ANTAGONISTS FOR TREATMENT OF CNS-RELATED DISORDERS AAPA B.V. (NL) 2015-05-14 WO disclosed