SCHEMBL1670425

SCHEMBL1670425

CCc1ccn(-c2c(C)noc2C)c1-c1ccc(OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
MAPT P10636 1/20 0.40
ALDH1A1 P00352 1/20 0.39
BRD4 O60885 7/20 0.39
BRD2 P25440 2/20 0.39
BRD3 Q15059 2/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670212 0.74 PTGS2 (0.44) PTGS2MAPTALDH1A1BRD4MEN1
SCHEMBL1672794 0.72 PTGS2 (0.44) PTGS2MAPTBRD4BRD2BRD3
SCHEMBL12987843 0.71 TUBB4A (0.40) PTGS2ALDH1A1BRD4BRD2BRD3
SCHEMBL12985937 0.71 TUBB4A (0.46) PTGS2MAPTALDH1A1BRD4
SCHEMBL12800447 0.68 PTGS2 (0.41) PTGS2MAPTALDH1A1BRD4BRD2
SCHEMBL12800962 0.68 PTGS2 (0.40) PTGS2MAPTBRD4
SCHEMBL12986522 0.67 TUBB4A (0.44) MAPTALDH1A1BRD4
SCHEMBL17833811 0.66 PTGS2 (0.72) PTGS2MAPTBRD4BRD2BRD3
SCHEMBL13195254 0.66 PTGS2 (0.41) PTGS2MAPTALDH1A1BRD4TDP1
SCHEMBL1672841 0.66 MAOA (0.39) PTGS2MAPTALDH1A1BRD4BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed