SCHEMBL1670212

SCHEMBL1670212

COc1ccc(-c2nccn2-c2c(C)noc2C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
BRD4 O60885 6/20 0.42
KDR P35968 1/20 0.42
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CREBBP Q92793 1/20 0.37
CHEK1 O14757 1/20 0.37
EGFR P00533 1/20 0.37
NTRK1 P04629 1/20 0.37
RET P07949 1/20 0.37
ROS1 P08922 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11771718 0.76 KDR (0.49) PTGS2KDRKDM4EMEN1ALDH1A1
SCHEMBL1672794 0.76 PTGS2 (0.44) PTGS2BRD4MAPTRAB9ASMN1; SMN2
SCHEMBL1670425 0.74 PTGS2 (0.41) PTGS2BRD4MAPTMEN1ALDH1A1
SCHEMBL1670708 0.74 PTGS2 (0.43) PTGS2BRD4MAPTLMNAKDM4E
SCHEMBL3270536 0.73 MAPK9 (0.51) PTGS2KDRMAPTKDM4EMEN1
SCHEMBL28186197 0.73 KDR (0.55) KDRKDM4EMEN1ALDH1A1HPGD
SCHEMBL1670909 0.71 PTGS2 (0.40) PTGS2BRD4MAPTKDM4EMEN1
SCHEMBL29975108 0.70 GLA (0.55) PTGS2KDRMAPTRAB9A
SCHEMBL28186123 0.70 GLA (0.55) PTGS2KDRMAPTRAB9A
SCHEMBL17484575 0.70 KDR (0.50) KDRMAPTKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed