SCHEMBL1670490

SCHEMBL1670490

Cc1noc(C)c1-c1c(-c2ccc(O)cc2F)cn(C)c1C(=N)NO

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 11/20 0.35
HSP90AB1 P08238 1/20 0.34
NSD3 Q9BZ95 1/20 0.34
ESR1 P03372 4/20 0.33
BCL2L1 Q07817 1/20 0.33
BAK1 Q16611 1/20 0.33
ESR2 Q92731 2/20 0.33
ERN1 O75460 1/20 0.33
CREBBP Q92793 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672810 0.84 BRD4 (0.40) BRD4HSP90AB1ERN1CREBBP
SCHEMBL1672792 0.83 ERN1 (0.38) BRD4NSD3BCL2L1BAK1ERN1
SCHEMBL1682601 0.83 HSP90AB1 (0.35) BRD4HSP90AB1NSD3ESR1BCL2L1
SCHEMBL1670492 0.82 BRD4 (0.35) BRD4HSP90AB1NSD3ESR1ESR2
SCHEMBL1672865 0.77 BRD4 (0.37) BRD4CREBBP
SCHEMBL21141736 0.76 GPBAR1 (0.37) BRD4HSP90AB1ESR1BCL2L1BAK1
SCHEMBL1682546 0.74 ESR1 (0.39) BRD4HSP90AB1ESR1ESR2
SCHEMBL1670808 0.73 TTR (0.34) ESR1ESR2
SCHEMBL1672899 0.71 ERN1 (0.38) BRD4BCL2L1BAK1ERN1CREBBP
SCHEMBL1671583 0.71 BRD4 (0.33) BRD4ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed