SCHEMBL16705452

SCHEMBL16705452

CCOC(=O)Cc1cc(I)no1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.42
VHL P40337 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751904 0.87 VHL (0.54) SMN1; SMN2VHLCA12CA1CA2
SCHEMBL26148033 0.81 ADRB2 (0.42) SMN1; SMN2VHLCA12CA1CA2
SCHEMBL25601889 0.79 KLK7 (0.41) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL19598756 0.78 PPARA (0.45) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL24348876 0.78 VHL (0.42) SMN1; SMN2VHLALDH1A1MAPTRAB9A
SCHEMBL25603628 0.76 PPARA (0.52) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL25602002 0.75 SMPD1 (0.47) SMN1; SMN2KDM4EALDH1A1
SCHEMBL24838097 0.75 SMPD1 (0.47) SMN1; SMN2KDM4EALDH1A1MEN1PKM
SCHEMBL25227460 0.74 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1MEN1MAPTHTT
SCHEMBL21159080 0.73 LMNA (0.43) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646446-B1 BROMODOMAIN INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2015-05-13 EP disclosed