SCHEMBL1670860

SCHEMBL1670860

Cn1c(Br)c(-c2ccc(O)cc2)c(I)c1C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.46
GRIA4 P48058 2/20 0.38
MMP3 P08254 1/20 0.37
SENP1 Q9P0U3 1/20 0.37
GAA P10253 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPK1 P28482 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ESR2 Q92731 2/20 0.33
MGAM O43451 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
CA12 O43570 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671716 0.82 GRIA2 (0.41) GRIA4GAAALDH1A1KDM4ELMNA
SCHEMBL12801011 0.80 SENP1 (0.36) ARSENP1GAAALDH1A1ALOX15
SCHEMBL1670503 0.73 AR (0.39) ARGRIA4MMP3SENP1GAA
SCHEMBL1670817 0.72 MLYCD (0.40) ARBRD4
SCHEMBL1670563 0.69 GRIA4 (0.39) ARGRIA4SENP1ALDH1A1KDM4E
SCHEMBL10591364 0.66 GRIA4 (0.42) ARGRIA4GAAALDH1A1MAPK1
SCHEMBL12800399 0.64 SENP1 (0.36) ARSENP1GAAALDH1A1ESR2
Acetonitrile SCHEMBL28239695 0.59 ESR1 (0.65) ARMMP3SENP1ALDH1A1KDM4E
SCHEMBL8873272 0.58 DYRK1A (0.30)
SCHEMBL1457230 0.58 ESR1 (0.71) MMP3SENP1ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed