SCHEMBL16712979

SCHEMBL16712979

Ic1cnccc1-c1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
KDM4E B2RXH2 6/20 0.48
LMNA P02545 3/20 0.48
METAP1 P53582 2/20 0.48
CCR1 P32246 2/20 0.48
CCR5 P51681 2/20 0.48
CCR8 P51685 2/20 0.48
CYP1A2 P05177 1/20 0.48
POLB P06746 1/20 0.48
BLM P54132 1/20 0.48
HIF1A Q16665 1/20 0.48
DOHH Q9BU89 1/20 0.48
P4HTM Q9NXG6 1/20 0.48
PRKCI P41743 1/20 0.45
TDO2 P48775 1/20 0.43
METAP2 P50579 2/20 0.42
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
TP53 P04637 3/20 0.42
TDP1 Q9NUW8 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19961428 0.85 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL277492 0.79 KDM4E (0.56) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL12854083 0.78 KDM4E (0.50) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL15787009 0.77 TDO2 (0.51) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL16897143 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL23598962 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL30343543 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL3034362 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL17180121 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1
SCHEMBL10205409 0.77 CYP2A6 (0.48) CYP2A6KDM4ELMNAMETAP1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069594-A1 GSK-3 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-05-14 WO disclosed