SCHEMBL16719320

SCHEMBL16719320

COC1=CC=CC(P(c2ccccc2)c2ccccc2)(P(c2ccccc2)c2ccccc2)C1c1ccccc1OC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.34
HTR2C P28335 3/20 0.33
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
ALDH1A1 P00352 4/20 0.33
MAPT P10636 4/20 0.33
KDM4E B2RXH2 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
USP2 O75604 1/20 0.33
GAA P10253 3/20 0.32
HPGD P15428 3/20 0.32
GLA P06280 2/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
ATM Q13315 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA7 P43166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6137738 1.00 HSD11B1 (0.34) HSD11B1HTR2CMEN1KMT2AALDH1A1
SCHEMBL6137485 0.85 MEN1 (0.36) HSD11B1HTR2CMEN1KMT2AALDH1A1
SCHEMBL8994728 0.67 GAA (0.34) MEN1KMT2AALDH1A1MAPTKDM4E
SCHEMBL5572903 0.66 MEN1 (0.32) HTR2CMEN1KMT2AL3MBTL1
1,2-Dimethoxybenzene SCHEMBL27452731 0.57 CA1 (0.93) KMT2AALDH1A1MAPTKDM4ESMN1; SMN2
SCHEMBL10571023 0.57 CA1 (0.48) HSD11B1HTR2CMEN1KMT2AALDH1A1
SCHEMBL1515163 0.56 HTR2C (0.75) HTR2CMEN1KMT2AATMCA12
SCHEMBL28829941 0.56 HTR2C (0.49) HSD11B1HTR2CMEN1KMT2AALDH1A1
SCHEMBL476857 0.55 CA1 (0.50) KMT2AALDH1A1SMN1; SMN2TP53MAPK1
SCHEMBL56425 0.55 CA1 (0.50) KMT2AALDH1A1SMN1; SMN2TP53MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068770-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINYLCYCLOPENTANE COMPOUNDS F. Hoffmann-La Roche AG (CH) 2016-09-21 EP disclosed
WO-2015073739-A1 PROCESSES FOR THE PREPARATION OF PYRIMIDINYLCYCLOPENTANE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2015-05-21 WO disclosed