SCHEMBL16719720

SCHEMBL16719720

Oc1c[c]ccc1-c1cncnc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ERN1 O75460 4/20 0.35
ATM Q13315 1/20 0.34
CYP2A6 P11509 1/20 0.32
AR P10275 2/20 0.31
PDK2 Q15119 1/20 0.30
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720501 0.81 CYP2A6 (0.48) CYP17A1CYP3A4CYP11B1CYP11B2ERN1
SCHEMBL16719697 0.80 CYP11B1 (0.42) CYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL16720179 0.78 QDPR (0.39) ERN1CCNCCDK8
SCHEMBL16720630 0.74 CYP11B1 (0.47) CYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL159940 0.74 ALDH1A1 (0.54) CYP2A6
SCHEMBL16719637 0.74 ESR1 (0.42) CYP3A4
SCHEMBL7945424 0.73 ATM (0.34) ERN1ATMCYP2A6PDK2
SCHEMBL10356483 0.71 ALDH1A1 (0.56) CYP17A1CYP3A4CYP11B1CYP11B2ATM
SCHEMBL9988102 0.71 BACE1 (0.38)
SCHEMBL16720203 0.71 ALOX5 (0.41) CYP3A4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed