SCHEMBL16719909

SCHEMBL16719909

Oc1c[c]ccc1-c1cccc(OC(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.43
ADORA2A P29274 1/20 0.43
THRA P10827 1/20 0.42
THRB P10828 1/20 0.42
P2RX1 P51575 1/20 0.39
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
XDH P47989 2/20 0.38
GALR1 P47211 1/20 0.38
DYRK1A Q13627 2/20 0.38
DHODH Q02127 1/20 0.37
KCNH2 Q12809 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
PTPN5 P54829 1/20 0.37
NPY5R Q15761 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319442 0.83 DRD1 (0.43) ADORA1THRATHRBDRD1KCNH2
SCHEMBL16720388 0.82 AURKA (0.39)
SCHEMBL2377419 0.81 HDAC4 (0.50) DYRK1A
SCHEMBL16719325 0.79 PTPN5 (0.47) ADORA1ADORA2ACTSSPTPN5
SCHEMBL361619 0.77 XDH (0.42) ADORA1ADORA2AXDHGALR1DYRK1A
SCHEMBL534246 0.77 SLC13A5 (0.44) ADORA1ADORA2AXDHGALR1DYRK1A
SCHEMBL2090977 0.75 THRA (0.50) ADORA1ADORA2ATHRATHRBP2RX1
SCHEMBL16720132 0.75 ESR2 (0.46) THRBPTPN5
SCHEMBL1274111 0.75 CYP1A1 (0.44) DYRK1ADHODH
SCHEMBL16719582 0.75 HSD17B1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed