SCHEMBL16719944

SCHEMBL16719944

COc1c[c]c(-c2cccc(F)c2)c(O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
PTGS1 P23219 1/20 0.39
MAOB P27338 1/20 0.39
NFE2L2 Q16236 2/20 0.39
ABL1 P00519 1/20 0.39
ABCB1 P08183 1/20 0.39
BCR P11274 1/20 0.39
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
FYN P06241 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
RELA Q04206 3/20 0.38
HDAC4 P56524 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
RPS6KB1 P23443 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720488 0.86 ABL1 (0.41) ESR2NPC1RAB9AABL1ABCB1
SCHEMBL16720142 0.83 BACE1 (0.46) NPC1RAB9AKDM4EALDH1A1ABL1
SCHEMBL16428843 0.75 CYP1A1 (0.53) ESR2NPC1RAB9AKDM4EALDH1A1
SCHEMBL4284645 0.75 KDM1A (0.42) ESR2NPC1RAB9AKDM4EALDH1A1
SCHEMBL16720127 0.74 COMT (0.40) ESR2NPC1RAB9AKDM4EALDH1A1
SCHEMBL16720157 0.73 ESR2 (0.50) ESR2PTGS1HSD17B1HSD17B2TRPM8
SCHEMBL16720131 0.71 ESR2 (0.47) ESR2NPC1RAB9APTGS1HSD17B1
SCHEMBL16720083 0.71 ESR2 (0.47) ESR2PTGS1HSD17B1HSD17B2FYN
SCHEMBL16720427 0.71 PDGFRB (0.45) NPC1RAB9AKDM4EALDH1A1PTGS1
SCHEMBL16719967 0.71 CYP1A1 (0.42) ESR2KDM4EALDH1A1FYNRELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed