SCHEMBL16720127

SCHEMBL16720127

COc1c[c]c(-c2ccncc2)c(O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.40
KDM4E B2RXH2 3/20 0.37
USP2 O75604 1/20 0.37
PDGFRB P09619 3/20 0.37
PDGFRA P16234 3/20 0.37
QDPR P09417 1/20 0.37
CYP1A2 P05177 4/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ERN1 O75460 1/20 0.36
CYP3A4 P08684 3/20 0.36
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MAPK1 P28482 2/20 0.36
RAB9A P51151 2/20 0.36
ABL1 P00519 1/20 0.36
ABCB1 P08183 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720142 0.83 BACE1 (0.46) KDM4EUSP2CYP1A2CYP3A4NPC1
SCHEMBL16720488 0.77 ABL1 (0.41) CYP1A2CYP1A1CYP1B1CYP3A4NPC1
SCHEMBL16719944 0.74 ESR2 (0.44) KDM4ENPC1SMN1; SMN2MAPK1RAB9A
SCHEMBL16720484 0.71 POLB (0.45) KDM4ECYP1A2CYP1A1CYP1B1CYP3A4
SCHEMBL16720143 0.70 MEN1 (0.51) CYP1A1CYP1B1MAPK1ABL1ABCB1
SCHEMBL16056542 0.69 CYP3A4 (0.48) KDM4EUSP2CYP1A1CYP1B1ERN1
SCHEMBL16720516 0.68 QDPR (0.36) KDM4EPDGFRBPDGFRAQDPRCYP1A2
SCHEMBL16720650 0.68 QDPR (0.36) PDGFRBPDGFRAQDPRERN1CYP3A4
SCHEMBL27934853 0.67 CYP3A4 (0.46) KDM4EUSP2CYP1A1CYP1B1ERN1
SCHEMBL16720286 0.67 PDGFRB (0.42) KDM4EUSP2PDGFRBPDGFRACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed