SCHEMBL16720157

SCHEMBL16720157

Oc1c[c]c(-c2cccc(F)c2)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
HSD17B1 P14061 3/20 0.44
HSD17B2 P37059 3/20 0.44
TAAR1 Q96RJ0 3/20 0.38
TRPM8 Q7Z2W7 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NR4A1 P22736 1/20 0.34
NR4A2 P43354 1/20 0.34
NR4A3 Q92570 1/20 0.34
NOTUM Q6P988 1/20 0.34
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720508 0.88 HSD17B1 (0.47) ESR2HSD17B1HSD17B2LMNA
SCHEMBL16720654 0.84 ESR1 (0.37) ESR2HSD17B1HSD17B2MAPTMEN1
SCHEMBL12488049 0.84 TAAR1 (0.41) ESR2HSD17B1HSD17B2TAAR1MAPT
SCHEMBL16720083 0.83 ESR2 (0.47) ESR2HSD17B1HSD17B2TAAR1TRPM8
SCHEMBL16720516 0.74 QDPR (0.36) ESR2MAPTLMNAALOX15NFKB1
SCHEMBL16719944 0.73 ESR2 (0.44) ESR2HSD17B1HSD17B2TRPM8PTGS1
SCHEMBL10494072 0.73 TAAR1 (0.41) ESR2HSD17B1HSD17B2TAAR1MAPT
SCHEMBL9646878 0.70 TAAR1 (0.39) ESR2HSD17B1HSD17B2TAAR1MEN1
SCHEMBL16720131 0.70 ESR2 (0.47) ESR2HSD17B1HSD17B2TAAR1PTGS1
SCHEMBL16719547 0.70 ESR2 (0.47) ESR2HSD17B1HSD17B2TAAR1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed