SCHEMBL16719989

SCHEMBL16719989

COc1cc(F)cc(-c2[c]cccc2O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
ABL1 P00519 5/20 0.37
ABCB1 P08183 5/20 0.37
BCR P11274 5/20 0.37
CYP3A4 P08684 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2A6 P11509 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP4B1 P13584 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP3A5 P20815 1/20 0.35
CYP2A7 P20853 1/20 0.35
CYP3A7 P24462 1/20 0.35
CYP2F1 P24903 1/20 0.35
CYP2C18 P33260 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719899 0.85 ABL1 (0.42) HDAC4HDAC8ABL1ABCB1BCR
SCHEMBL2377417 0.80 HDAC4 (0.55) HDAC4HDAC8ABL1ABCB1BCR
SCHEMBL16719521 0.80 HSD17B1 (0.40) CYP3A4KDM1A
SCHEMBL17514939 0.78 CYP1A1 (0.46) ABL1ABCB1BCRCYP3A4CYP1A1
SCHEMBL16719654 0.78 KDM4E (0.47) HDAC4HDAC8HDAC2
SCHEMBL16719996 0.77 ALOX5 (0.35) PGR
SCHEMBL16720629 0.77 CYP11B1 (0.44) HDAC4HDAC8CYP3A4CYP1A1CYP1A2
SCHEMBL16719852 0.76 ALDH1A1 (0.36) HDAC4HDAC8ABL1ABCB1BCR
SCHEMBL16720131 0.74 ESR2 (0.47)
SCHEMBL9650164 0.72 NPC1 (0.35) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed