SCHEMBL16720101

SCHEMBL16720101

Oc1cccc(-c2ccn[c]n2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 13/20 0.52
HSD17B2 P37059 12/20 0.52
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 2/20 0.45
METAP2 P50579 1/20 0.45
CYP19A1 P11511 2/20 0.42
PIK3CA P42336 1/20 0.40
CYP17A1 P05093 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
ESR1 P03372 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
ESR2 Q92731 1/20 0.39
FYN P06241 1/20 0.39
CDC7 O00311 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15477525 0.79 KMO (0.45) CYP19A1
SCHEMBL11107619 0.79 METAP2 (0.45) METAP2
SCHEMBL16720064 0.79 KMO (0.45) CYP3A4CYP17A1CYP11B1CYP11B2ESR2
SCHEMBL557899 0.77 KMT2A (0.41) METAP2
SCHEMBL3654046 0.71 CYP1A2 (0.47) CYP2C9CYP19A1CYP17A1CYP11B1CYP11B2
SCHEMBL989535 0.70 CYP2A6 (0.52) CYP3A4CYP2C9METAP2CYP19A1CYP1A2
SCHEMBL30862097 0.70 HSD17B1 (0.66) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL1899480 0.69 HSD17B1 (0.58) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL20566349 0.69 HSD17B1 (0.58) HSD17B1HSD17B2CYP3A4CYP2C9METAP2
SCHEMBL17626014 0.69 KMO (0.49) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed