SCHEMBL1672802

SCHEMBL1672802

CC(=O)Oc1ccc(-c2ncc(C#N)n2-c2c(C)noc2C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.39
LMNA P02545 3/20 0.39
TSHR P16473 2/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
TP53 P04637 4/20 0.36
NPC1 O15118 2/20 0.36
PKM P14618 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 3/20 0.35
CREBBP Q92793 2/20 0.35
MAPT P10636 1/20 0.34
GAPDH P04406 1/20 0.34
THRB P10828 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
BRD2 P25440 1/20 0.32
MAOB P27338 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670909 0.68 PTGS2 (0.40) RAB9ASMN1; SMN2BRD4MAPTHSD17B10
SCHEMBL1670700 0.65 ERN1 (0.40) BRD4CREBBPBRD2
SCHEMBL11611224 0.65 HSD17B10 (0.50) RAB9ALMNATSHRNFKB1NFKB2
SCHEMBL11759468 0.65 HSD17B10 (0.50) RAB9ALMNATSHRNFKB1NFKB2
SCHEMBL11755257 0.64 HSD17B10 (0.53) RAB9ALMNATSHRNFKB1NFKB2
Water SCHEMBL9344643 0.62 HSD17B10 (0.73) RAB9ALMNATSHRNFKB1NFKB2
SCHEMBL27751423 0.62 LMNA (0.49) RAB9ALMNATSHRNFKB1NFKB2
SCHEMBL5945230 0.62 HSD17B10 (0.58) LMNATP53PKMMAPTTHRB
SCHEMBL25284190 0.62 HSD17B10 (0.50) RAB9ALMNATSHRNFKB1NFKB2
SCHEMBL11750060 0.61 HSD17B10 (0.49) RAB9ALMNATSHRNFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed