Bicarbonate

Bicarbonate

SCHEMBL16735545

CCc1ccc([C@@H](C(=O)Nc2cccc(CC3CC3)c2)[C@@H](C)C(F)(F)F)cc1.O=C(O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
ACKR3 P25106 3/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
PARP1 P09874 1/20 0.40
GCGR P47871 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
FAAH O00519 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9899621 1.00 SMN1; SMN2 (0.42) SMN1; SMN2ACKR3TP53MAPTPARP1
Bicarbonate SCHEMBL16735655 0.91 FAAH (0.44) ACKR3FAAHHTR1AHTR1DHTR1B
Bicarbonate SCHEMBL16735564 0.90 ACKR3 (0.47) ACKR3FAAHALDH1A1CCR3
Bicarbonate SCHEMBL9900300 0.90 ALDH1A1 (0.43) SMN1; SMN2ACKR3MAPTFAAHALDH1A1
Bicarbonate SCHEMBL16735571 0.90 NLRP3 (0.41) ACKR3ALDH1A1HTR1AHTR1DHTR1B
Bicarbonate SCHEMBL16735613 0.86 S1PR1 (0.49) ACKR3MAPTFAAHMEN1KMT2A
Bicarbonate SCHEMBL16735611 0.84 KLKB1 (0.35) SMN1; SMN2MAPTPARP1ALDH1A1UBE2M
SCHEMBL10006523 0.84 MAPT (0.40) SMN1; SMN2ACKR3TP53MAPTPARP1
SCHEMBL9899617 0.84 MAPT (0.40) SMN1; SMN2ACKR3TP53MAPTPARP1
SCHEMBL9899772 0.83 HDAC3 (0.40) SMN1; SMN2ACKR3TP53MAPTPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed