Bicarbonate

Bicarbonate

SCHEMBL16735655

Cc1ccc(C(C(=O)Nc2cccc(CC3CC3)c2)C(C)C(F)(F)F)cc1.O=C(O)O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.44
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
ACKR3 P25106 3/20 0.41
HTR1A P08908 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
KLKB1 P03952 1/20 0.38
DRD2 P14416 1/20 0.38
CCR3 P51677 3/20 0.38
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL9899621 0.91 SMN1; SMN2 (0.42) FAAHACKR3HTR1AHTR1DHTR1B
Bicarbonate SCHEMBL16735545 0.91 SMN1; SMN2 (0.42) FAAHACKR3HTR1AHTR1DHTR1B
Bicarbonate SCHEMBL16735564 0.91 ACKR3 (0.47) FAAHACKR3DRD2CCR3
Bicarbonate SCHEMBL9900300 0.91 ALDH1A1 (0.43) FAAHACKR3CCR3
Bicarbonate SCHEMBL16735613 0.89 S1PR1 (0.49) FAAHACKR3
Bicarbonate SCHEMBL16735571 0.89 NLRP3 (0.41) ACKR3HTR1AHTR1DHTR1B
SCHEMBL10006265 0.84 MAPT (0.38) ACKR3DRD2
SCHEMBL9899892 0.83 MAPT (0.38) ACKR3DRD2
Bicarbonate SCHEMBL3702662 0.81 ACHE (0.41) ACKR3CCR3
Bicarbonate SCHEMBL3696258 0.81 KCNJ6 (0.39) ACKR3KLKB1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed