Bicarbonate

Bicarbonate

SCHEMBL16735546

C[C@H]([C@H](C(=O)Nc1cc(CC2CC2(F)F)ccc1Cl)c1ccc(Cl)cc1)C(F)(F)F.O=C(O)O

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 1/20 0.39
TRPV1 Q8NER1 1/20 0.37
PANK3 Q9H999 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
FFAR2 O15552 7/20 0.35
ALDH1A1 P00352 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
LMNA P02545 1/20 0.34
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
IDO1 P14902 2/20 0.33
TDO2 P48775 2/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL16735616 0.89 KMT2A (0.41) KMT2AL3MBTL1MEN1TRPV1PANK3
SCHEMBL10006239 0.84 KMT2A (0.39) KMT2AL3MBTL1MEN1TRPV1PANK3
SCHEMBL10006324 0.82 KMT2A (0.41) KMT2AL3MBTL1MEN1TRPV1PANK3
Bicarbonate SCHEMBL9899636 0.82 KMT2A (0.41) KMT2AL3MBTL1MEN1TRPV1PANK3
SCHEMBL1932029 0.82 KMT2A (0.41) KMT2AL3MBTL1MEN1TRPV1PANK3
Bicarbonate SCHEMBL16735635 0.81 KMT2A (0.47) KMT2AL3MBTL1MEN1SMN1; SMN2ALDH1A1
Bicarbonate SCHEMBL16735627 0.81 FFAR2 (0.38) FFAR2CYP3A4
SCHEMBL14805608 0.81 KMT2A (0.40) KMT2AL3MBTL1MEN1TRPV1PANK3
SCHEMBL14798044 0.81 KMT2A (0.40) KMT2AL3MBTL1MEN1TRPV1PANK3
SCHEMBL6903201 0.81 L3MBTL1 (0.45) KMT2AL3MBTL1MEN1TRPV1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed