Bicarbonate

Bicarbonate

SCHEMBL16735669

C[C@H]([C@H](C(=O)Nc1cc(CC2CC2)ccc1Cl)c1ccc(Cl)cc1F)C(F)(F)F.O=C(O)O

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 1/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
OPRL1 P41146 2/20 0.35
TRPV1 Q8NER1 1/20 0.35
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL16735616 0.87 KMT2A (0.41) PANK3KMT2AMEN1L3MBTL1PDK1
Bicarbonate SCHEMBL16735568 0.86 KMT2A (0.39) PANK3KMT2AMEN1L3MBTL1TRPV1
SCHEMBL1933212 0.85 MEN1 (0.42) PANK3KMT2AMEN1L3MBTL1PDK1
SCHEMBL10006505 0.85 KMT2A (0.38) PANK3KMT2AMEN1L3MBTL1DPP4
Bicarbonate SCHEMBL16735627 0.83 FFAR2 (0.38) TP53UBE2MDCUN1D1
Bicarbonate SCHEMBL9899636 0.82 KMT2A (0.41) PANK3KMT2AMEN1L3MBTL1TRPV1
SCHEMBL1932886 0.82 L3MBTL1 (0.38) PANK3KMT2AMEN1L3MBTL1PDK1
Bicarbonate SCHEMBL16735635 0.81 KMT2A (0.47) KMT2AMEN1L3MBTL1SMN1; SMN2HPGD
SCHEMBL1932882 0.80 L3MBTL1 (0.38) KMT2AMEN1L3MBTL1PDK1PDK2
Bicarbonate SCHEMBL16735610 0.80 CCR3 (0.36) TRPV1TP53MAPTUBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed