SCHEMBL16748705

SCHEMBL16748705

CCCCOc1cc(-c2nc(C(=O)O)co2)[n+](O)cc1OCCCC

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.37
S1PR3 Q99500 1/20 0.35
XDH P47989 3/20 0.34
CNR2 P34972 1/20 0.34
PTPN11 Q06124 1/20 0.33
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
WDR5 P61964 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16748703 0.90 DAGLA (0.34) TP53KDM4ENPC1ALDH1A1RAB9A
SCHEMBL9915358 0.88 S1PR3 (0.37) TP53S1PR3XDHPTPN11WDR5
SCHEMBL9915354 0.79 TP53 (0.33) TP53S1PR3PDE4BPDE4D
SCHEMBL16748687 0.79 HPGD (0.43) CNR2NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9915503 0.78 TP53 (0.39) TP53S1PR3XDHPTPN11KDM4E
SCHEMBL17040094 0.77 HDAC1 (0.46) CNR2PTPN11KDM4EALDH1A1SMN1; SMN2
SCHEMBL16747529 0.77 XDH (0.41) TP53XDHCNR2WDR5ALDH1A1
SCHEMBL17244012 0.74 S1PR1 (0.41) XDHPTPN11
SCHEMBL2874377 0.74 CYP1A2 (0.46) CNR2PTPN11KDM4EALDH1A1SMN1; SMN2
SCHEMBL16748641 0.74 GAA (0.43) TP53S1PR3XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed