SCHEMBL16752102

SCHEMBL16752102

CNCC(CCCN)N(C)C

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.30
CHRM2 P08172 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16752067 0.86 OPRD1 (0.31)
SCHEMBL557874 0.78 PRMT3 (0.37) TDP1
SCHEMBL9385386 0.78 OPRD1 (0.33)
SCHEMBL20835084 0.77 ALDH1A1 (0.40)
SCHEMBL22872239 0.77
SCHEMBL571022 0.77 CHRM2 (0.35) TDP1CHRM2
SCHEMBL13397769 0.75 OPRD1 (0.36)
SCHEMBL14392136 0.75 OPRD1 (0.32)
SCHEMBL8851759 0.75 CHRM2 (0.33) TDP1CHRM2
SCHEMBL16752028 0.73 OPRD1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2878609-B1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND TOSOH CORP (JP) 2019-06-05 EP claimed
US-20150203727-A1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND TOSOH CORPORATION (JP) 2015-07-23 US claimed
EP-2878609-A1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND Tosoh Corporation (JP) 2015-06-03 EP claimed
EP-2878609-B1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND TOSOH CORP (JP) 2019-06-05 EP disclosed
US-9777199-B2 Amine catalyst for curing polyisocyanate compound and polyisocyanate adhesive composition containing amine catalyst for curing polyisocyanate compound TOSOH CORPORATION (JP) 2017-10-03 US disclosed
US-20150203727-A1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND TOSOH CORPORATION (JP) 2015-07-23 US disclosed
EP-2878609-A1 AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND AND POLYISOCYANATE ADHESIVE COMPOSITION CONTAINING AMINE CATALYST FOR CURING POLYISOCYANATE COMPOUND Tosoh Corporation (JP) 2015-06-03 EP disclosed