SCHEMBL1677263

SCHEMBL1677263

CC(C)Oc1cc(Oc2ccc(S(C)(=O)=O)cn2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
GCK P35557 9/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
POLB P06746 2/20 0.38
KCNH2 Q12809 1/20 0.37
CHRNA7 P36544 1/20 0.37
TP53 P04637 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ACACB O00763 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1038221 0.83 ALDH1A1 (0.43) ALDH1A1GCKPOLB
SCHEMBL12734099 0.81 KDM4E (0.43) ALDH1A1POLBKDM4EACACB
SCHEMBL1677258 0.80 MMP2 (0.44) ALDH1A1ALOX5APFEN1POLBKCNH2
SCHEMBL12807181 0.80 KDM4E (0.39) ALDH1A1POLBKDM4EACACB
SCHEMBL1677111 0.80 CA12 (0.42) ALDH1A1PTGS1PTGS2ACACB
SCHEMBL14994793 0.77 G6PD (0.50) GCKPOLBKCNH2PTGS1PTGS2
SCHEMBL563822 0.77 GCK (0.41) GCKALOX5APFEN1PTGS1PTGS2
SCHEMBL15449639 0.76 ALDH1A1 (0.69) ALDH1A1GCKKCNH2CHRNA7PTGS1
SCHEMBL12807214 0.76 GCK (0.41) ALDH1A1GCKPTGS1PTGS2
SCHEMBL12807211 0.74 GCK (0.39) ALDH1A1GCKALOX5APFEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8673942-B2 Fused ring compounds and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-03-18 US disclosed
US-8673942-B2 Fused ring compounds and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-03-18 US disclosed
US-20110098297-A1 FUSED RING COMPOUNDS AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-04-28 US disclosed
WO-2009125873-A1 FUSED RING COMPOUNDS AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110098297-A1 FUSED RING COMPOUNDS AND USE THEREOF GCKR, GPR119, SLC5A1 ALDH1A1 305/4885GCK 4/4885ALOX5AP 3657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.