SCHEMBL16784653

SCHEMBL16784653

CN1C2C1C21Cc2ccc(OCCNS(=O)(=O)c3cnn(C)c3)cc2C1Cc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 13/20 0.51
HTR1A P08908 4/20 0.39
HTR7 P34969 4/20 0.39
KCNH2 Q12809 1/20 0.39
DGAT1 O75907 1/20 0.35
MGAT3 Q09327 1/20 0.35
MGAT2 Q10469 1/20 0.35
DRD2 P14416 2/20 0.34
HTR6 P50406 2/20 0.34
SLC8A1 P32418 1/20 0.34
ADRA1D P25100 1/20 0.33
HTR2A P28223 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
ALK Q9UM73 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229752 0.92 SLC6A9 (0.52) SLC6A9HTR1AHTR7KCNH2SLC8A1
SCHEMBL16784630 0.91 SLC6A9 (0.54) SLC6A9HTR1AHTR7KCNH2
SCHEMBL16784632 0.91 SLC6A9 (0.52) SLC6A9HTR1AHTR7KCNH2HTR6
SCHEMBL16229753 0.90 SLC6A9 (0.41) SLC6A9HTR1AHTR7DGAT1MGAT3
SCHEMBL16229789 0.88 DGAT1 (0.40) SLC6A9DGAT1MGAT3MGAT2
SCHEMBL16229749 0.87 SLC6A9 (0.55) SLC6A9KCNH2
SCHEMBL16784654 0.86 POLB (0.40) SLC6A9HTR1AHTR7SLC8A1ALK
SCHEMBL16229806 0.84 DGAT1 (0.35) SLC6A9DGAT1MGAT3MGAT2HTR6
SCHEMBL16784626 0.83 SLC6A9 (0.50) SLC6A9HTR1AHTR7KCNH2DRD2
SCHEMBL16784639 0.83 SLC6A9 (0.45) SLC6A9HTR1AHTR7KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed