SCHEMBL167878

SCHEMBL167878

COc1ccc(CN(Cc2ccc(OC)cc2)C(=S)NC(=O)c2cccc(Cl)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
MEN1 O00255 4/20 0.67
KMT2A Q03164 4/20 0.67
TDP1 Q9NUW8 2/20 0.67
ALOX12 P18054 2/20 0.67
HTT P42858 2/20 0.67
NPSR1 Q6W5P4 2/20 0.67
L3MBTL1 Q9Y468 2/20 0.67
GPR55 Q9Y2T6 1/20 0.67
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
CYP2D6 P10635 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2C19 P33261 2/20 0.60
PKM P14618 1/20 0.58
MAPT P10636 1/20 0.52
LMNA P02545 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
BCL2A1 Q16548 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165611 0.90 ALDH1A1 (0.72) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL168734 0.87 ALDH1A1 (0.69) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL12467306 0.87 ALDH1A1 (0.72) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL256654 0.86 ALDH1A1 (0.67) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL168039 0.86 ALDH1A1 (0.67) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL167636 0.86 ALDH1A1 (0.77) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL168699 0.86 ALDH1A1 (0.90) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL1542223 0.86 PKM (0.63) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL168012 0.85 ALDH1A1 (0.69) ALDH1A1MEN1KMT2ATDP1ALOX12
SCHEMBL168590 0.84 ALDH1A1 (0.64) ALDH1A1MEN1KMT2ATDP1ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed