SCHEMBL1679330

SCHEMBL1679330

COc1ccc(-c2cncc(C(C)C(=O)O)c2C)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.49
CYP2C19 P33261 1/20 0.49
MMP2 P08253 1/20 0.46
MMP3 P08254 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP12 P39900 1/20 0.46
MMP13 P45452 1/20 0.46
MMP14 P50281 1/20 0.46
MMP16 P51512 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
CHEK1 O14757 1/20 0.44
SLC22A12 Q96S37 3/20 0.43
MAP4K4 O95819 2/20 0.41
PTGS2 P35354 3/20 0.40
PTGS1 P23219 2/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
CDC42 P60953 1/20 0.40
RAC1 P63000 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1679080 0.82 MMP2 (0.55) APPCYP2C19MMP2MMP3MMP9
SCHEMBL1679633 0.75 CYP2C19 (0.54) APPCYP2C19MMP2MMP3MMP9
SCHEMBL5266001 0.74 CYP11B1 (0.48) MMP2MMP3MMP9MMP8MMP12
Hydrochloric Acid SCHEMBL4808141 0.70 PTGS2 (0.54) PTGS2PTGS1AKR1C3AKR1C2CDC42
SCHEMBL1679541 0.70 PTGS2 (0.45) CYP2C19MAP4K4PTGS2CYP1A2
SCHEMBL1679164 0.70 ERN1 (0.42) CYP2C19SLC22A12MAP4K4PTGS2CYP1A2
SCHEMBL1678493 0.70 PTGS2 (0.67) APPCYP2C19MMP2MMP3MMP9
SCHEMBL6372641 0.67 PTGS2 (0.57) APPCYP2C19MMP2MMP3MMP9
SCHEMBL7960349 0.67 PTGS2 (0.57) PTGS2PTGS1AKR1C3AKR1C2CDC42
SCHEMBL350067 0.67 PTGS2 (0.71) APPCYP2C19PTGS2PTGS1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7923573-B2 Benzene compound having 2 or more substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-04-12 US disclosed
US-20080004301-A1 Benzene Compound Having 2 or More Substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004301-A1 Benzene Compound Having 2 or More Substituents NR1H2, NR1H3, NCOR2 APP 1870/4885CYP2C19 238/4885MMP2 4839/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.