SCHEMBL1679541

SCHEMBL1679541

COc1ccc(-c2cncc(Br)c2C)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.45
KMT2A Q03164 3/20 0.44
ACVR1 Q04771 2/20 0.43
MAOB P27338 1/20 0.43
MAPT P10636 1/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
RPS6KA3 P51812 1/20 0.41
QPCT Q16769 1/20 0.41
QPCTL Q9NXS2 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
PLK4 O00444 1/20 0.40
AURKA O14965 1/20 0.40
DYRK3 O43781 1/20 0.40
MAP4K4 O95819 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1891962 0.81 MAPT (0.49) PTGS2KMT2AMAPTCYP11B1CYP11B2
SCHEMBL28198658 0.79 PTGS2 (0.41) PTGS2KMT2AACVR1MAPTCYP11B1
SCHEMBL24500005 0.79 MAPK14 (0.38) KMT2AMAPTRPS6KA3CYP1A2CYP3A4
SCHEMBL30530579 0.79 MAPK14 (0.38) KMT2AMAPTRPS6KA3CYP1A2CYP3A4
SCHEMBL954335 0.78 LMNA (0.39) KMT2AMAPTRPS6KA3AURKACDK1
SCHEMBL20999462 0.78 ALDH1A1 (0.45) MAOBRPS6KA3CYP1A2CYP2B6PLK4
SCHEMBL29597422 0.78 ALDH1A1 (0.45) MAOBRPS6KA3CYP1A2CYP2B6PLK4
SCHEMBL1679164 0.76 ERN1 (0.42) PTGS2KMT2AACVR1MAPTCYP11B1
SCHEMBL28912340 0.75
SCHEMBL6173237 0.72 CYP11B1 (0.45) PTGS2KMT2AMAPTCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7923573-B2 Benzene compound having 2 or more substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-04-12 US disclosed
US-20080004301-A1 Benzene Compound Having 2 or More Substituents DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-03 US disclosed
EP-1806332-A1 BENZENE COMPOUND HAVING 2 OR MORE SUBSTITUENTS Daiichi Sankyo Company, Limited (JP) 2007-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004301-A1 Benzene Compound Having 2 or More Substituents NR1H2, NR1H3, NCOR2 PTGS2 3493/4885KMT2A 2190/4885ACVR1 901/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.