SCHEMBL16795443

SCHEMBL16795443

Cc1cc(NC2CCN(C(=O)O)CC2)cc(C)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.44
CYP3A4 P08684 3/20 0.44
PHGDH O43175 2/20 0.41
SIGLEC9 Q9Y336 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21590380 0.88 NOS2 (0.40) ROCK2CYP3A4PHGDHSIGLEC9KDM4E
SCHEMBL21606962 0.81 ALDH1A1 (0.62) KDM4EMAPT
SCHEMBL4693278 0.78 MAPT (0.51) KDM4ELMNANPSR1MAPT
SCHEMBL17303596 0.78 GBA1 (0.54) ROCK2CYP3A4MAPT
SCHEMBL15829881 0.77 MAPT (0.45) ROCK2CYP3A4MAPT
SCHEMBL5969516 0.77 EPHX2 (0.54) CYP3A4KDM4ELMNANPSR1
SCHEMBL3801054 0.76 SPR (0.50) KDM4EMAPT
SCHEMBL3900029 0.75 ALDH1A1 (0.48) KDM4EUSP2NPSR1HSD17B10MAPT
SCHEMBL16111210 0.75 OPRM1 (0.60) NOS3NOS1NOS2OPRM1
SCHEMBL13860480 0.75 MAPT (0.45) SIGLEC9KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed