SCHEMBL168028

SCHEMBL168028

NC(Cc1ccc(O)cc1)C(=O)OS(=O)(=O)OC(=O)C(N)Cc1ccc(O)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.59
TAAR1 Q96RJ0 3/20 0.46
SLC6A2 P23975 1/20 0.46
HDAC8 Q9BY41 2/20 0.46
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
DPP4 P27487 1/20 0.42
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
ERAP2 Q6P179 1/20 0.40
LNPEP Q9UIQ6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29969329 0.91 SLC7A5 (0.53) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL6523945 0.89 SLC7A5 (0.57) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL168029 0.89 SLC7A5 (0.57) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL29969049 0.88 SLC7A5 (0.50) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL25234890 0.87 SLC7A5 (0.56) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL3476198 0.87 SLC7A5 (0.56) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL4453960 0.82 SLC7A5 (0.67) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL27680265 0.82 SLC7A5 (0.67) SLC7A5TAAR1SLC6A2HDAC8ESR1
SCHEMBL27725763 0.82 SLC7A5 (0.54) SLC7A5TAAR1HDAC8ALPIPKM
SCHEMBL8012238 0.81 SLC7A5 (0.65) SLC7A5TAAR1SLC6A2HDAC8ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10059739-B2 Non-benzenoid aromatic systems for imaging, monitoring and therapy MEDIBEACON INC. (US) 2018-08-28 US disclosed
US-20160083426-A1 NON-BENZENOID AROMATIC SYSTEMS FOR IMAGING, MONITORING AND THERAPY MEDIBEACON INC. (US) 2016-03-24 US disclosed
US-9226980-B2 Azulene and azaazulene systems for imaging, monitoring and therapy MEDIBEACON INC. (US) 2016-01-05 US disclosed
US-9186349-B2 Diaza heterocyclic compounds for phototherapy MALLINCKRODT LLC (US) 2015-11-17 US disclosed
US-8731655-B2 Compounds containing acyclic N-N bonds for phototherapy MALLINCKRODT LLC (US) 2014-05-20 US disclosed
US-20120289884-A1 Fused Ring Diarylamino Photosensitizers for Phototherapy MALLINCKRODT LLC (US) 2012-11-15 US disclosed
US-20120203102-A1 AZULENE AND AZAAZULENE SYSTEMS FOR IMAGING, MONITORING AND THERAPY MALLINCKRODT LLC (US) 2012-08-09 US disclosed
US-20120058954-A1 Diaza Heterocyclic Compounds for Phototherapy OCERA THERAPEUTICS LLC 2012-03-08 US disclosed
US-20120053511-A1 Compounds Containing Acyclic N-N Bonds for Phototherapy MALLINCKRODT BRAND PHARMACEUTICALS LLC (F/K/A MALLINCKRODT BRAND PHARMACEUTICALS, INC.) 2012-03-01 US disclosed
US-20110288033-A1 Disulfide Compounds for Phototherapy MALLINCKRODT INC. (US) 2011-11-24 US disclosed
US-20110264026-A1 Azo Derivatives and Uses Thereof in Phototherapy MALLINCKRODT LLC 2011-10-27 US disclosed
WO-2011084571-A2 AZIDE DERIVATIVES FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2011-07-14 WO disclosed
WO-2011060113-A1 SULFENAMIDE COMPOUNDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2011-05-19 WO disclosed
WO-2011031915-A2 NON-BENZENOID AROMATIC SYSTEMS FOR IMAGING, MONITORING AND THERAPY MALLINCKRODT INC. (US) 2011-03-17 WO disclosed
WO-2010132525-A1 COMPOUNDS CONTAINING ACYCLIC N-O BONDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-11-18 WO disclosed
WO-2010132554-A2 DIAZA HETEROCYCLIC COMPOUNDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-11-18 WO disclosed
WO-2010132547-A2 OXAZA HETEROCYCLIC COMPOUNDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-11-18 WO disclosed
WO-2010132515-A1 COMPOUNDS CONTAINING ACYCLIC N-N BONDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-11-18 WO disclosed
EP-2227474-A1 AZO AND DIAZA DERIVATIVES AND USES THEREOF IN PHOTOTHERAPY Mallinckrodt Inc. (US) 2010-09-15 EP disclosed
WO-2010060018-A1 AZO AND DIAZA DERIVATIVES AND USES THEREOF IN PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-05-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288033-A1 Disulfide Compounds for Phototherapy SPIN1, QSOX1, SAV1 SLC7A5 1450/4885TAAR1 3060/4885SLC6A2 3362/4885
US-20110264026-A1 Azo Derivatives and Uses Thereof in Phototherapy IRAK1, IL1A, MALT1 SLC7A5 4004/4885TAAR1 4076/4885SLC6A2 4874/4885
US-20120058954-A1 Diaza Heterocyclic Compounds for Phototherapy BAD, BID, CASP3 SLC7A5 3999/4885TAAR1 4775/4885SLC6A2 4419/4885
US-20120203102-A1 AZULENE AND AZAAZULENE SYSTEMS FOR IMAGING, MONITORING AND THERAPY AZI2, ALK, ZKSCAN2 SLC7A5 726/4885TAAR1 491/4885SLC6A2 2159/4885
US-20160083426-A1 NON-BENZENOID AROMATIC SYSTEMS FOR IMAGING, MONITORING AND THERAPY PAH, AHR, ALK SLC7A5 1091/4885TAAR1 779/4885SLC6A2 728/4885
US-10059739-B2 Non-benzenoid aromatic systems for imaging, monitoring and therapy PAH, AHR, ALK SLC7A5 1091/4885TAAR1 779/4885SLC6A2 728/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.